{"entity": "publication", "iuid": "0f1760ea3e0c48a1bb18e9eafc1c7412", "timestamp": "2026-06-08T10:33:07.306Z", "links": {"self": {"href": "https://publications-affiliated.scilifelab.se/publication/0f1760ea3e0c48a1bb18e9eafc1c7412.json"}, "display": {"href": "https://publications-affiliated.scilifelab.se/publication/0f1760ea3e0c48a1bb18e9eafc1c7412"}}, "title": "A Synthesis of \"Dual Warhead\" \u03b2-Aryl Ethenesulfonyl Fluorides and One-Pot Reaction to \u03b2-Sultams.", "authors": [{"family": "Chinthakindi", "given": "Praveen K", "initials": "PK"}, {"family": "Govender", "given": "Kimberleigh B", "initials": "KB"}, {"family": "Kumar", "given": "A Sanjeeva", "initials": "AS"}, {"family": "Kruger", "given": "Hendrik G", "initials": "HG"}, {"family": "Govender", "given": "Thavendran", "initials": "T"}, {"family": "Naicker", "given": "Tricia", "initials": "T"}, {"family": "Arvidsson", "given": "Per I", "initials": "PI"}], "type": "journal article", "published": "2017-02-03", "journal": {"title": "Org. Lett.", "issn": "1523-7060", "volume": "19", "issue": "3", "pages": "480-483", "issn-l": "1523-7052"}, "abstract": "Herein, we report an operationally simple, ligand- and additive-free oxidative boron-Heck coupling that is compatible with the ethenesulfonyl fluoride functional group. The protocol proceeds at room temperature with chemoselectivity and E-isomer selectivity and offers facile access to a wide range of \u03b2-aryl/heteroaryl ethenesulfonyl fluorides from commercial boronic acids. Furthermore, we demonstrate a \"one-pot click\" reaction to directly transform the products to aryl-substituted \u03b2-sultams.", "doi": "10.1021/acs.orglett.6b03634", "pmid": "28075600", "labels": {"Affiliated researcher": null}, "xrefs": [], "notes": [], "created": "2018-12-05T11:05:13.684Z", "modified": "2018-12-05T11:05:13.706Z"}